Manufacturer: TEVA
Pharmaceutical name: Tamoxifen Citrate
Pack: 1 pack (30 tabs (10 mg))
Tamoxifen is a potent Selective Estrogen Receptor Modulator (SERM), often categorized as an anti-estrogen. Intriguingly, while it acts as an antagonist, it can also function as an agonist by mimicking estrogen in certain areas of the body, while exerting anti-estrogen effects in others. Being one of the earliest SERMs available, it remains widely prescribed in medicine. Additionally, tamoxifen is utilized by anabolic steroid users, though it is not classified as an anabolic steroid itself—something that often leads to confusion regarding its role in steroid cycles. Tamoxifen is fundamentally a SERM, making it an important component for bodybuilders.
Shortly after anabolic steroid users recognized the significance of this compound, they began using it as an anti-estrogen during steroid cycles to mitigate estrogen-related side effects. Tamoxifen is also commonly employed in Post Cycle Therapy (PCT) recovery plans, which is arguably its most beneficial application for steroid users.
For breast cancer patients, the drug's effects are clear-cut. By blocking estrogen from binding, it prevents the cancer from leveraging the hormone for its sustenance.
Regarding anabolic steroid users, Tamoxifen's main role during steroid cycles is to prevent gynecomastia. It does not seem to significantly counteract water retention, another common estrogenic effect, although there are other methods to manage this issue. When it comes to gynecomastia prevention, Tamoxifen can be sufficient for many men and should be the primary option if effective. If it fails, a more powerful Aromatase Inhibitor, such as Arimidex (Anastrozole), may be necessary. However, Aromatase Inhibitors can adversely affect cholesterol levels. While their individual effects may not be significantly negative, combining them with aromatizing steroids appears to exacerbate cholesterol issues. Though Aromatase Inhibitors can help control cholesterol, if Tamoxifen can do the job, it should be the first choice, especially since it has a positive impact on cholesterol levels.
Another notable benefit for bodybuilders using Tamoxifen is its capacity to enhance natural testosterone production. Even though it primarily functions as an anti-estrogen, it also has strong testosterone-stimulating properties. Tamoxifen can obstruct the